High-Purity Testolone – Precisely formulated RAD-140 solution suspended in PEG-400 for consistent solubility and accuracy.
Verified Quality – Each batch undergoes independent third-party testing to confirm purity and concentration.
Secure and Convenient Ordering – Sports Technology Labs accepts credit card payments for a smooth and reliable checkout experience.
Liquid RAD-140
High-Quality Liquid RAD-140 For Sale
Sports Technology Labs provides high-purity RAD-140 for sale for laboratory use. RAD-140, commonly known as Testolone, is a selective androgen receptor modulator (SARM) investigated for its selective interaction with androgen receptors in muscle and bone tissues. It should not be confused with its esterified form, RAD-150, also known as TLB-150.
RAD-140 binds to the androgen receptors (AR) selectively and does not produce the full range of androgenic effects as similar substances like testosterone, DHT, or anabolic steroids. This product is supplied strictly as a research chemical; it is not FDA approved, not for human consumption, and not intended to diagnose, treat, cure, or prevent any disease.
Independent Lab-Tested: RAD-140 Certificate of Analysis
At Sports Technology Labs, transparency and quality assurance are non-negotiable. A third-party, ISO-accredited laboratory rigorously tests every batch of our Liquid RAD-140 (Testolone) to verify identity, purity, and concentration.
This ensures you’re receiving a research-grade product that meets the highest standards. All results are batch-specific and linked directly to the product you receive.
RAD-140 FAQs
A study performed in 2010 found that after 28 days of testing RAD-140, the testosterone levels in all three groups were suppressed to approximately 200−300 ng/dL, with similar suppression in all groups. However, testosterone levels were significantly different for only the 0.01 mg/kg group (p < 0.05).
Although it is not known to be particularly androgenic, there is little available information regarding the safety profile of RAD-140 in female test subjects, and females should be cautious with participating in clinical research with RAD-140 until more information is available.
While it is not known to be particularly androgenic on its own, RAD-140 administration can free testosterone that is otherwise bound to SHBG in the male body, and this can indirectly increase the risk of hair loss.
RAD-140 is a selective androgen receptor modulator (SARM) studied for its potential to increase muscle mass and strength while minimizing side effects associated with anabolic steroids. It is strictly intended for laboratory and research use, and this information has not been tested in human trials.
Yes, every batch undergoes third-party testing to verify identity, purity (≥99%), and concentration. You can view the certificate of analysis above.
Both forms contain the same active compound, and all SARMs start as raw powder regardless of final delivery method. The choice largely depends on your priorities:
Choose Liquid if: You want convenience, potentially faster absorption, and precise measuring control. Choose Powder if: You want the most cost-effective option and are willing to prepare it yourself with proper lab equipment.
It’s essential, whichever form you decide on, to ensure that you’ve chosen a reputable source providing SARMs of the highest purity, verified by independent lab testing.
No. RAD-140 is a research chemical with an unapproved status. It is not FDA approved and is not sold for human consumption.
RAD-140 is a selective androgen receptor modulator designed to preferentially engage receptors in muscle and bone tissues, potentially limiting effects in other tissues. Risks remain; long-term human safety data are limited.
Signals include liver toxicity (e.g., cholestatic injury), testosterone suppression, possible lipid changes (lower HDL, higher LDL), and reports of mood disturbance or sleep disruption; long-term effects are not well characterized. RAD-140 is prohibited in sport by WADA.
Prioritize reputable suppliers offering third-party testing (COAs), consistent labeling and packaging with tamper-evident features, detailed product descriptions, secure checkout, and transparent business details. Avoid counterfeit or substandard products by purchasing from reliable vendors that comply with regulatory standards.
Legal status varies by jurisdiction. Researchers must review legal considerations, local laws, and institutional policies before purchase. The World Anti-Doping Agency bans RAD-140 for competitive athletes (source). Some regions impose age restrictions for purchase.
Post-cycle therapy is sometimes discussed in non-clinical, anecdotal contexts due to potential testosterone suppression. No PCT regimen is approved for RAD-140; Sports Technology Labs does not provide guidance on human use and follows all FDA regulations surrounding the product. This product is not for human use.
Products are shipped in discreet packaging with clear research-use labeling. Our platform uses encrypted processing to protect financial information.
Why is Sports Technology Labs the best place to buy RAD-140 online?
Research-grade formulation: Precisely formulated liquid Testolone, suspended for consistent solubility and accurate measurement.
Testing & transparency: ISO-accredited third-party testing with batch-linked COAs.
Compliance-first: Clear research-use labeling, discreet packaging, and rigorous safety standards.
Trusted operations: Established reputable vendors, practices, secure payments, and responsive support.
A recent study involving chemical analyses of 44 different products sold and marketed as SARMs on the internet revealed that quality control in this industry varies significantly from one company to the next.
Only 52% of the products tested contained the product advertised, 59% contained amounts that differed from the label, a shocking 39% contained other unapproved drugs, 25% contained substances not listed on the label, and 9% contained no active substance at all. It is critical when performing research with SARMs to only purchase the highest quality, verified by third-party analysis.
Many websites offer RAD-140 for sale, but Sports Technology Labs is the best place to buy RAD-140 online because of their consistent, verifiable, high-quality products, safer bottling and packaging, fast shipping, and excellent customer service. The internet seems to be full of sites offering Testolone and related substances. This may leave you wondering which of these many options you should select.
Some websites are more interested in making quick cash than in ensuring that their customers receive dependable products. That’s why you need to buy only from websites with established quality-control procedures.
When you buy SARMs from Sports Technology Labs, you are choosing the highest quality ingredients. Minimum 98% pure compounds tested and certified by accredited American third-party labs, suspended in USP-grade (the highest grade) PEG-400, bottled in America.
Our products come in glass bottles with fixed glass droppers to prevent the leaching of unwanted plasticizers like BPA and extend shelf life, and to avoid contamination between uses with external measuring tools.
We run a transparent business, with no discreet payment methods necessary and no misrepresentation of our products, only the highest quality research chemicals available online, secured by our 60-day money-back guarantee. For orders totaling $149 or more, we offer free shipping. If you’re in a hurry to receive your products, we also provide express shipping options.
Additionally, customers who sign up for our email list receive a 10% discount and an additional 10% off when paying with cryptocurrency. When you choose Sports Technology Labs, you are choosing the best place to buy RAD-140. Our RAD-140 is also available in pure powder form.
We are also committed to offering first-rate customer service. You’re always welcome to contact us with any questions or concerns you have about our RAD-140.
Additional information
Weight
3.0 oz
RAD-140 / Testolone
All Sports Technology Labs SARMs are third-party tested by MZ Biolabs, an independent laboratory based in Arizona. Each batch is bottled and tested in the USA to ensure accuracy and purity. Our Certificates of Analysis confirm that products meet the listed specifications:
RAD-140 is a non-steroidal agent designed to engage androgen receptors in target tissues preferentially. In preclinical settings, RAD-140 has been explored for effects related to anabolic activity in muscle and bone, with a pharmacology that is unlike anabolic steroids due to its tissue selectivity. Studies also examine potential neuroprotective effects through pathways associated with neuronal cell survival. Evidence in humans remains limited; ongoing research continues to evaluate safety, pharmacokinetics, and translational relevance.
Mechanism of Action: Androgen Receptors, Muscle and Bone
As a selective androgen receptor modulator, RAD-140 binds androgen receptors with high affinity in muscle cells and bone tissues. Downstream signaling in preclinical models has included increases in protein synthesis, support of lean muscle mass and muscle fiber hypertrophy, and markers relevant to bone density. Because of its selectivity for target tissues, RAD-140 is frequently contrasted with anabolic steroids that may influence a broader range of other tissues. Its tissue selectivity profile and receptor pharmacodynamics remain active areas of investigation.
In Vitro, the RAD-140 SARM has produced a wide array of effects, including:
Increased weight loss and body fat loss
Increased lean muscle growth and protein synthesis
Increased removal of beta-amyloid plaques from the brain
Increased protection against breast and prostate cancer
Increased endurance
However, it is essential to note that the Food and Drug Administration (FDA) has not confirmed any health effects of RAD-140 in humans or approved it for human use; therefore, the drug should be used in a laboratory setting.
High AR Binding Affinity of RAD-140
RAD-140 demonstrated excellent affinity for the AR (Ki = 7 nM), higher even than DHT and most anabolic steroids. For reference, the affinity for the androgen receptor (AR) for testosterone in a recent preclinical model was 29 nM, and 10 nM for DHT.
Unlike testosterone and most other AR-mediated anabolic agents, Testolone is orally bioavailable, so it does not require injection for proper absorption, and it is considered by many researchers to be one of the best SARMs for bulking and adding lean body mass.
Testolone is a relatively recent addition to the list of SARMs for sale; it was developed in 2010 as a possible treatment for osteoporosis and muscle gains. More recent testing performed on rats and primates, as well as clinical trials, has indicated that it may provide additional benefits.
Research Applications (Preclinical and Early Clinical Context)
Muscle biology: Studies exploring pathways linked to lean muscle growth, hypertrophy, and anabolic signaling in skeletal muscle.
Bone health: Investigation of androgen-receptor–mediated effects on bone turnover and potential support of bone density.
Neuroprotection: Evaluation of cell survival signaling and anti-apoptotic markers in neuronal models, with preclinical reports of neuroprotective effects.
Oncology research: Assessment in select hormone-receptor–positive cancer models for anti-proliferative activity.
Important: Findings above are based primarily on non-human or early-phase research. RAD-140 is not approved for therapeutic use, not for human consumption, and remains a research-only material.
Side Effects of RAD-140
While RAD-140 and other SARMs do not cause androgenic side effects to the same extent as anabolic steroids like testosterone, reports have revealed the potential for nausea, aggression, reduction in natural testosterone levels, or mild male pattern hair loss from the use of RAD-140. A single-member case report indicated drug-induced liver injury after 11 months of the use of an antidepressant, as well as intermittent use of RAD-140 and LGD-4033.
The limitations of this study, however, are that it includes only one test subject, 11 months of concurrent antidepressant use, the quality and quantity of SARMs used by the subject were not monitored, and additional comorbidities were not investigated.
Several case reports exist indicating the potential for selective androgen receptor modulators to contribute to liver injury but none involve a significant sample size or test controls to date. Like other SARMs, RAD-140 may trigger a negative feedback loop and a reduction in natural testosterone production and testicle size though further research is needed to determine the likelihood and severity of this occurrence.
RAD-140 and Muscle Growth
A study on young male cynomolgus monkeys investigated the anabolic effects of 28 days of RAD-140 at a dosage of 0.01mg/kg, 0.1mg/kg, and 1mg/kg per day. A mean weight gain of 10% was observed in both the 0.1mg/kg/day group and the 1mg/kg/day group, indicating a quantity response curve that leveled off and provided no additional benefit with higher quantities.
There was no consistent effect on body fat mass in either group; however, muscle mass increased in the 0.1 and 1mg/kg/day groups. No significant increases in liver enzymes or prostate weight were reported in either group, suggesting a high level of selectivity for androgen receptors in muscle tissue.
RAD-140 and Neuroprotection
Androgens have shown clinical significance in preventing neuronal apoptosis and improving cognitive function in Alzheimer’s Disease (AD), primarily through a nongenomic mechanism of the Androgen Receptor (AR). Rapid phosphoinositide 3-kinase/Akt signaling, activated by androgens, regulates the expression of proteins linked to apoptosis such as Bax, Seladin 1, survivin, XIAP, and Bcl-xl.
Androgens can also maintain the integrity of neurons and thus improve cognitive function. Studies have shown that Aβ impairs the synaptic structure and function of hippocampal neurons, which is reversed by androgen administration, resulting in improved cognitive performance in AD animal models. Although the underlying exact mechanisms are not yet fully understood, androgen’s action of inhibiting Aβ-induced apoptosis appears to play a role.
RAD–140 and Cellular Protection
A 2014 study investigated the neuroprotective effects of RAD-140 on cultured neurons and male rats that were lesioned with kainate. The experiment included two parts: one in vitro, involving cell cultures, and another in vivo, through animal testing.
Results from the in vitro study showed that RAD-140 was able to prevent cell death and restore mitochondrial membrane potential, indicating that it could offer neuroprotection much like testosterone and other androgens investigated for these effects.
The in vivo experiment tested the efficacy of RAD-140 on male rats with kainate-induced seizures and showed a significant reduction in seizure activity compared to controls.
RAD-140 and Dementia
Another study on rats found that RAD-140 had neuroprotective benefits of a kind that may prevent Alzheimer’s disease and similar disorders, and may be safer than conventional testosterone therapy The group treated with 3 mg/kg RAD-140 was able to replicate the same level of muscle tissue growth as the group treated with 1 mg/kg testosterone, with about half of the androgenic activity in the prostate.
RAD-140 and Breast Cancer
A 2017 study investigated the effects of RAD-140 on breast cancer cells. The study evaluated the efficacy of RAD-140 in inhibiting the growth of breast cancer cells that were positive for both androgen receptors (ARs) and estrogen receptors (ERs).
Results showed that in in vivo and in vitro models of AR/ER+ breast cancer, RAD-140 was able to significantly reduce the growth and metastases of breast cancer cells without disrupting their cell cycle, indicating it could be a promising therapy for treating such cancers.
Moreover, the study also showed that RAD-140 had distinct mechanisms of action from those of anti-estrogens and aromatase inhibitors, which suggests that it could provide an additional therapeutic approach to treating hormone-sensitive breast cancers.
Overall, this study suggests that RAD-140 could be a potential option for AR/ER-positive breast cancer. Still, more data are needed to determine its safety relative to other methods currently used.
Product Data
CAS Number: 1182367-47-0
Formula: C20H16ClN5O2
Molar Mass: 393.83 g/mol
Half-life: 44.7 hours
Class: Selective androgen receptor modulator
Storage: Store in a cool, dry place away from direct sunlight to maximize shelf life.
30 mL Liquid RAD-140 per bottle with 15 milligrams per milliliter.
Includes a graduated 1 mL glass pipette for convenient measurement.
Glass bottle with UV resistance to minimize degradation.
Tamper-proof seal to ensure safety in transit.
Less than 5% variance in concentration, guaranteeing consistency.
Formulated and packaged to prevent evaporation in storage.
SKU: 6
This preparation is for laboratory research purposes only and is not approved by the FDA for human consumption. RAD–140/Testolone IS NOT A DIETARY OR SPORTS SUPPLEMENT.
Abuse Warning
RAD-140 is an investigational compound still awaiting FDA approval and is not a dietary supplement. At Sports Technology Labs, we are chemical suppliers, not medical doctors, and our expertise is sourcing and quality control. Sports Technology Labs does not encourage or condone consumer use of SARMs products; they are for research purposes only.
SARMs should only be used under the supervision and direction of a medical doctor or designated research authority. We strongly discourage the use of SARMs for performance enhancement in sports and bodybuilding, and warn against “bro science” and peer consensus when making decisions about human health.
Safety, Risks, and Legal Considerations
Unapproved status: RAD-140 is not an approved drug product; regulatory agencies (e.g., FDA) do not approve it for human consumption. The World Anti-Doping Agency prohibits SARM use in competitive sport. The long-term safety profile remains unknown.
Potential risks observed:
Liver toxicity: Case reports have described cholestatic liver injury and jaundice associated with RAD-140 exposure.
Testosterone suppression: Suppression of endogenous testosterone has been observed; post-cycle therapy is sometimes discussed in non-clinical contexts, though no regimen is approved for RAD-140 by the FDA.
Lipids and mood: Reports include mood changes (irritability, restlessness), sleep disturbance, and adverse lipid profile changes (lower HDL, higher LDL).
Unknown long-term effects: Human safety data are limited; caution is warranted.
Legal considerations: Distribution, possession, or sale may be restricted depending on jurisdiction. Researchers are responsible for compliance with local laws, applicable laws, and institutional policies. RAD-140 is provided by Sports Technology Labs solely for research purposes. Some regions impose age restrictions on purchase; laws are subject to change.
Quality Assurance: Avoiding Counterfeit or Substandard Products
The research chemical marketplace can include counterfeit or substandard products, counterfeit or contaminated products, and unsafe products distributed by unverified online vendors. Independent testing in the SARM category has identified mislabeling, incorrect dosage strength, and undeclared actives in some products. Authenticity safeguards include:
Third-party testing: Every batch undergoes independent analysis for identity, purity, and concentration; third-party testing results (COAs) are made available.
Product authenticity and labeling: Clear labeling, consistent packaging, tamper-evident seals, and detailed product descriptions to support traceability and product quality.
Vendor verification:Reputable vendors provide transparent business information, secure checkout, and responsive support. Customer feedback can help assess supplier reliability.
Regulatory awareness: Be mindful of limited oversight and verify that suppliers operate within relevant regulatory standards.
To avoid counterfeit purchases, researchers should prioritize vendors with verifiable COAs, transparent practices, and compliance with industry regulations. STL sources from reputable manufacturers and operates as a reliable vendor for research materials.
Scientific References:
1. Miller, C. P., Shomali, M., Lyttle, C. R., O’Dea, L. S., Herendeen, H., Gallacher, K., Paquin, D., Compton, D. R., Sahoo, B., Kerrigan, S. A., Burge, M. S., Nickels, M., Green, J. L., Katzenellenbogen, J. A., Tchesnokov, A., & Hattersley, G. (2010). Design, Synthesis, and Preclinical Characterization of the Selective AR Modulator (SARM) RAD-140. ACS medicinal chemistry letters, 2(2), 124–129.
2. Jayaraman, A., Christensen, A., Moser, V. A., Vest, R. S., Miller, C. P., Hattersley, G., & Pike, C. J. (2014). Selective AR modulator RAD-140 is neuroprotective in cultured neurons and kainate-lesioned male rats. Endocrinology, 155(4), 1398–1406.
3. D. K. Hamson, S. R. Wainwright, J. R. Taylor, B. A. Jones, N. V. Watson, L. A. M. Galea, Androgens Increase Survival of Adult-Born Neurons in the Dentate Gyrus by an Androgen Receptor-Dependent Mechanism in Male Rats, Endocrinology, Volume 154, Issue 9, 1 September 2013, Pages 3294–3304
4. Yu, Ziyang et al. “Selective Androgen Receptor Modulator RAD-140 Inhibits the Growth of Androgen/Estrogen Receptor–Positive BC Models with a Distinct Mechanism of Action.” MK 677 Clinical Cancer Research 23 (2017): 7608 – 7620.
5. LoRusso P, Hamilton E, Ma C, Vidula N, Bagley RG, Troy S, Annett M, Yu Z, Conlan MG, Weise A. A First-in-Human Phase 1 Study of a Novel Selective AR Modulator (SARM), RAD-140, in ER+/HER2- Metastatic BC. Clin Br Cancer. 2022 Jan;22(1):67-77. doi: 10.1016/j.clbc.2021.08.003. Epub 2021 Aug 20. PMID: 34565686.
6. Puskas, J. (2022). Pre-clinical assessment of the selective androgen receptor modulator RAD–140 to increase muscle mass and bone mineral density (Doctoral dissertation).
7. Flores JE, Chitturi S, Walker S. Drug-Induced Liver Injury by Selective Androgenic Receptor Modulators. Hepatol Commun. 2020 Jan 3;4(3):450-452. doi: 10.1002/hep4.1456. PMID: 32140660; PMCID: PMC7049679.
8. Bing L, Wu J, Zhang J, Chen Y, Hong Z, Zu H. DHT inhibits the Aβ25-35-induced apoptosis by regulation of seladin-1, survivin, XIAP, bax, and bcl-xl expression through a rapid PI3-K/Akt signaling in C6 glial cell lines. Neurochem Res. 2014;40(1):41–48.
9. Huo DS, Sun JF, Zhang B, Yan XS, Wang H, Jia JX, Yang ZJ. Protective effects of testosterone on cognitive dysfunction in Alzheimer’s disease model rats induced by oligomeric beta amyloid peptide 1–42. J Toxicol Environ Health A. 2016;79(19):856–863.
10. Van Wagoner RM, Eichner A, Bhasin S, Deuster PA, Eichner D. Chemical Composition and Labeling of Substances Marketed as Selective Androgen Receptor Modulators and Sold via the Internet. JAMA. 2017 Nov 28;318(20):2004-2010. doi: 10.1001/jama.2017.17069. Erratum in: JAMA. 2018 Feb 20;319(7):724. PMID: 29183075; PMCID: PMC5820696.
